Catalog_no
|
BDMC0039
|
Product_name
|
Trametinib (GSK-1120212)
|
Category
|
抑制剂与激动剂
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Size
|
10mg/50mg/100mg
|
Price
|
560.00/880.00/1320.00
|
Specificity
|
Target: MEK. Fields: GSK1120212 (JTP-74057, trametinib) is a highly specific and potent MEK1 and MEK2 inhibitor with IC50 of 0.92 nM and 1.8 nM, respectively.
|
Dilution
|
IC50: 2 nM (MEK1/2)[1]
|
Purification
|
>98%
|
Concentration
|
靶点:MEK;IC50: 2 nM (MEK1/2)[1]
|
Storage_stability
|
2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
|
othername
|
GSK212, GSK 1120212 , JTP-74057, trametinib, GSK1120212
|
Observed_band
|
615.39
|
Notes
|
GSK1120212 (JTP-74057, trametinib) is a highly specific and potent MEK1 and MEK2 inhibitor with IC50 of 0.92 nM and 1.8 nM, respectively.
|